5GN5ABCD

Crystal structure of glycerol kinase from trypanosoma brucei gambiense complexed with cumarin derivative-17
Link type Probability Loop ranges Chain A piercings Chain B piercings Chain C piercings Chain D piercings
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
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Other Other 36% -A +511B +511B +67C +331C -353C +377C -389C +423C -512D -512A -376D -511D
Interpreting sequences
Chain A Sequence
ATMKYVGSIDQGTTSTRFIIFDERQRPVSVHQVPHTQHTPHPGWLEHDPMEIFRSACKCMSVAIAKLRQKDASFRKIEAIGITNQRETTVAWDRVTKEPLCYAPVWNDLRTYDITKKVTAELGGGDSMFASKITGLPVSTYFAAFKMRWMLENVPAVADACRRGTLCFGTIDTWLMYKLSGGKAFVTDVTNASRTFLMDLRTRKWSPELCEKLKIPMETLPEIRSNSELFGYVETDECGVAAALNERTPIMGSIGDQQSALFGNMCFEKGEAKNTYGTGCFLLMNVGEEARFSKHGLLSTVGFQVGRDGPCYYALEGAIACAGATVEWMRRNMNLFSHITECEKLARSVPGTQGIVFVPAFSGLLAPYWDPSARGTIVGMTLKTTRAHVIRAALQAIALQLNDVVGSMKRDAGLNLSSLRVDGGLSKNGLLMEIQASLLGVDILVPSMHETTALGAALCAGLAAGVWTSLEEVKAVSRRENSWKTVSPSGSAMEREAMIAEWREALKRTKWAK
Chain A Sequence
ATMKYVGSIDQGTTSTRFIIFDERQRPVSVHQVPHTQHTPHPGWLEHDPMEIFRSACKCMSVAIAKLRQKDASFRKIEAIGITNQRETTVAWDRVTKEPLCYAPVWNDLRTYDITKKVTAELGGGDSMFASKITGLPVSTYFAAFKMRWMLENVPAVADACRRGTLCFGTIDTWLMYKLSGGKAFVTDVTNASRTFLMDLRTRKWSPELCEKLKIPMETLPEIRSNSELFGYVETDECGVAAALNERTPIMGSIGDQQSALFGNMCFEKGEAKNTYGTGCFLLMNVGEEARFSKHGLLSTVGFQVGRDGPCYYALEGAIACAGATVEWMRRNMNLFSHITECEKLARSVPGTQGIVFVPAFSGLLAPYWDPSARGTIVGMTLKTTRAHVIRAALQAIALQLNDVVGSMKRDAGLNLSSLRVDGGLSKNGLLMEIQASLLGVDILVPSMHETTALGAALCAGLAAGVWTSLEEVKAVSRRENSWKTVSPSGSAMEREAMIAEWREALKRTKWAK
Chain A Sequence
ATMKYVGSIDQGTTSTRFIIFDERQRPVSVHQVPHTQHTPHPGWLEHDPMEIFRSACKCMSVAIAKLRQKDASFRKIEAIGITNQRETTVAWDRVTKEPLCYAPVWNDLRTYDITKKVTAELGGGDSMFASKITGLPVSTYFAAFKMRWMLENVPAVADACRRGTLCFGTIDTWLMYKLSGGKAFVTDVTNASRTFLMDLRTRKWSPELCEKLKIPMETLPEIRSNSELFGYVETDECGVAAALNERTPIMGSIGDQQSALFGNMCFEKGEAKNTYGTGCFLLMNVGEEARFSKHGLLSTVGFQVGRDGPCYYALEGAIACAGATVEWMRRNMNLFSHITECEKLARSVPGTQGIVFVPAFSGLLAPYWDPSARGTIVGMTLKTTRAHVIRAALQAIALQLNDVVGSMKRDAGLNLSSLRVDGGLSKNGLLMEIQASLLGVDILVPSMHETTALGAALCAGLAAGVWTSLEEVKAVSRRENSWKTVSPSGSAMEREAMIAEWREALKRTKWAK
Chain A Sequence
ATMKYVGSIDQGTTSTRFIIFDERQRPVSVHQVPHTQHTPHPGWLEHDPMEIFRSACKCMSVAIAKLRQKDASFRKIEAIGITNQRETTVAWDRVTKEPLCYAPVWNDLRTYDITKKVTAELGGGDSMFASKITGLPVSTYFAAFKMRWMLENVPAVADACRRGTLCFGTIDTWLMYKLSGGKAFVTDVTNASRTFLMDLRTRKWSPELCEKLKIPMETLPEIRSNSELFGYVETDECGVAAALNERTPIMGSIGDQQSALFGNMCFEKGEAKNTYGTGCFLLMNVGEEARFSKHGLLSTVGFQVGRDGPCYYALEGAIACAGATVEWMRRNMNLFSHITECEKLARSVPGTQGIVFVPAFSGLLAPYWDPSARGTIVGMTLKTTRAHVIRAALQAIALQLNDVVGSMKRDAGLNLSSLRVDGGLSKNGLLMEIQASLLGVDILVPSMHETTALGAALCAGLAAGVWTSLEEVKAVSRRENSWKTVSPSGSAMEREAMIAEWREALKRTKWAK
sequence length 513,513,513,513
structure length 513,513,513,513
publication title Discovery of trypanocidal coumarins with dual-inhibition for African trypanosomes glycerol kinase and alternative oxidase
rcsb
molecule tags Transferase
molecule keywords Glycerol kinase
source organism Trypanosoma brucei gambiense
pdb deposition date2016-07-19
LinkProt deposition date2017-08-29
Image from the rcsb pdb (www.rcsb.org)
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LinkProt | Interdisciplinary Laboratory of Biological Systems Modelling